Synthesis of 1,2,3-triazolylpyranosides through click chemistry reaction
نویسندگان
چکیده
منابع مشابه
Synthesis of phenyl-adducted cyclodextrin through the click reaction
a Plant Polymer Research Unit, National Center for Agricultural Utilization Research, USDA/Agricultural Research Services, 1815 N. University Street, Peoria, IL 61604, USA Ashland Hercules Water Technologies, 500 Hercules Road, Wilmington, DE 19808-1599, USA Mycotoxin Research Unit, National Center for Agricultural Utilization Research, USDA/Agricultural Research Services, 1815 N. University St...
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Targeting small molecules to diseased tissues as therapy or diagnosis is a significant challenge in drug delivery. Drug-eluting devices implanted during invasive surgery allow the controlled presentation of drugs at the disease site, but cannot be modified once the surgery is complete. We demonstrate that bioorthogonal click chemistry can be used to target circulating small molecules to hydroge...
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Click chemistry is an approach that uses efficient and reliable reactions, such as Cu(I)-catalyzed azide-alkyne cycloaddition (CuAAC), to bind two molecular building blocks. CuAAC has broad applications in medicinal chemistry and other fields of chemistry. This review describes the general features and applications of CuAAC in solid-phase synthesis (CuAAC-SP), highlighting the suitability of th...
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ژورنال
عنوان ژورنال: Tetrahedron Letters
سال: 2012
ISSN: 0040-4039
DOI: 10.1016/j.tetlet.2012.01.102